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Pharmaceutical Nutrient Depletion

Writer: Olga BrennanOlga Brennan

Updated: Feb 25

In this post, I have compiled a list of commonly prescribed drugs and their resultant vitamin deficiencies. As you may suspect, the side effects of most common drugs emerge from the nutrient depletion caused by them. Organ systems pay a toll in order to expel, degrade and process foreign substances. It is very common to end up treating side effects of drugs with more and more drugs, which leads to deeper, more severe nutrient loss.


Mechanisms of Depletion: Nutrients may be depleted through various mechanisms, such as reduced absorption (e.g., PPIs lowering stomach acid), increased excretion (e.g., diuretics flushing out minerals), interference with metabolism (e.g., statins inhibiting CoQ10 synthesis), or disruption of gut microbiota (e.g., antibiotics affecting vitamin production).


Drug Class

Examples

Nutrients Depleted

Statins

Atorvastatin, Simvastatin, Rosuvastatin

Coenzyme Q10 (CoQ10), Vitamin D

Proton Pump Inhibitors (PPIs)

Omeprazole, Esomeprazole, Pantoprazole

Vitamin B12, Magnesium, Calcium, Iron, Vitamin C

H2 Receptor Antagonists

Ranitidine, Famotidine

Vitamin B12, Calcium, Iron, Vitamin D

Diuretics (Loop)

Furosemide, Bumetanide

Potassium, Magnesium, Calcium, Zinc, Vitamin B1 (Thiamine), Vitamin B6, Vitamin C

Diuretics (Thiazide)

Hydrochlorothiazide, Chlorthalidone

Potassium, Magnesium, Zinc, Sodium, Folic Acid

Diuretics (Potassium-Sparing)

Spironolactone, Amiloride

Folic Acid, Calcium

ACE Inhibitors

Lisinopril, Enalapril, Captopril

Zinc, Sodium

Beta Blockers

Metoprolol, Atenolol, Propranolol

Coenzyme Q10, Melatonin, Chromium

Antidepressants (SSRIs)

Sertraline, Fluoxetine, Citalopram

Folic Acid, Sodium, Vitamin B6

Antidepressants (Tricyclics)

Amitriptyline, Nortriptyline

Coenzyme Q10, Vitamin B2 (Riboflavin), Sodium

Antipsychotics

Quetiapine, Risperidone, Olanzapine

Vitamin D, Folic Acid, Vitamin B12

Mood Stabilizers

Lithium

Folic Acid, Inositol

Oral Hypoglycemics

Metformin

Vitamin B12, Coenzyme Q10, Folic Acid

Antibiotics (Broad-Spectrum)

Amoxicillin, Ciprofloxacin, Doxycycline

Biotin, Vitamins B1, B2, B3, B5, B6, B12, Vitamin K, Magnesium, Calcium, Probiotics

Corticosteroids

Prednisone, Hydrocortisone, Fluticasone

Calcium, Vitamin D, Magnesium, Potassium, Zinc, Vitamin B6, Vitamin C, Selenium

Oral Contraceptives

Ethinylestradiol combinations

Folic Acid, Vitamins B2, B6, B12, Vitamin C, Magnesium, Zinc, Coenzyme Q10, Tyrosine

NSAIDs

Ibuprofen, Naproxen, Aspirin

Folic Acid, Vitamin C, Iron, Glutathione

Opioids

Hydrocodone, Oxycodone, Morphine

Folic Acid, Vitamin C, Iron, Potassium

Anticonvulsants

Phenytoin, Carbamazepine, Valproate

Folic Acid, Vitamin D, Vitamin B12, Calcium, Vitamin K, Biotin

Benzodiazepines

Diazepam, Lorazepam, Alprazolam

Melatonin, Calcium, Magnesium

Stimulants

Methylphenidate, Amphetamine (Adderall)

Magnesium, Zinc

Bisphosphonates

Alendronate, Risedronate

Calcium, Magnesium, Vitamin D

Antiretrovirals

Zidovudine, Efavirenz

Vitamin B12, Vitamin D, Zinc, Magnesium

Chemotherapy Agents

Methotrexate, Cisplatin

Folic Acid, Magnesium, Potassium, Vitamin B12 (varies by agent)

The following table lists the effects of each nutrient deficiency:

Nutrient

Symptoms of Deficiency

Biotin (Vitamin B7)

Hair loss, brittle nails, skin rashes (especially around the mouth), fatigue, depression, neurological symptoms (e.g., numbness, tingling)

Calcium

Muscle cramps, spasms, osteoporosis, brittle bones, tooth decay, numbness or tingling, irregular heartbeat

Chromium

Impaired glucose tolerance (leading to blood sugar issues), fatigue, weight loss, nerve damage

Coenzyme Q10 (CoQ10)

Fatigue, muscle weakness, heart problems (e.g., palpitations, heart failure), high blood pressure, cognitive decline

Folic Acid (Vitamin B9)

Fatigue, weakness, anemia (megaloblastic), shortness of breath, irritability, mouth sores, neural tube defects in pregnancy

Glutathione

Increased oxidative stress, fatigue, weakened immune system, muscle weakness, neurological issues

Inositol

Mood disorders (e.g., anxiety, depression), insomnia, hair loss, skin issues

Iron

Fatigue, weakness, pale skin, anemia, shortness of breath, brittle nails, cold hands/feet, dizziness

Magnesium

Muscle cramps, fatigue, irritability, irregular heartbeat, nausea, weakness, migraines, poor sleep

Melatonin

Insomnia, difficulty falling/staying asleep, daytime fatigue, mood changes

Potassium

Muscle weakness, cramps, fatigue, irregular heartbeat (arrhythmias), constipation, tingling/numbness

Probiotics (Gut Flora)

Digestive issues (e.g., bloating, diarrhea, constipation), weakened immunity, mood changes (via gut-brain axis)

Selenium

Fatigue, hair loss, weakened immune system, muscle weakness, cognitive decline

Sodium

Nausea, headache, confusion, fatigue, muscle cramps, seizures (severe cases)

Tyrosine

Fatigue, depression, difficulty concentrating, low motivation, impaired thyroid function

Vitamin B1 (Thiamine)

Fatigue, muscle weakness, confusion, memory loss, nerve damage (e.g., tingling), heart issues (e.g., beriberi)

Vitamin B2 (Riboflavin)

Mouth sores, cracked lips, sore throat, fatigue, sensitivity to light, skin rashes

Vitamin B3 (Niacin)

Fatigue, depression, skin rashes (pellagra), diarrhea, headache, memory loss

Vitamin B5 (Pantothenic Acid)

Fatigue, irritability, muscle cramps, numbness/tingling, digestive issues

Vitamin B6 (Pyridoxine)

Anemia, depression, confusion, weakened immunity, skin rashes, nerve issues (e.g., tingling, neuropathy)

Vitamin B12 (Cobalamin)

Fatigue, weakness, anemia, numbness/tingling, memory loss, depression, balance issues

Vitamin C

Fatigue, scurvy (bleeding gums, bruising), slow wound healing, joint pain, weakened immunity

Vitamin D

Bone pain, muscle weakness, osteoporosis, fatigue, depression, impaired immunity

Vitamin K

Easy bruising, excessive bleeding, poor blood clotting, weak bones

Zinc

Weakened immunity, hair loss, slow wound healing, loss of taste/smell, skin rashes, diarrhea

Additional Notes:

  1. Overlap in Symptoms: Many nutrient deficiencies share symptoms like fatigue, weakness, and irritability because these nutrients often work together in metabolic pathways (e.g., B vitamins in energy production).

  2. Severity: Mild deficiencies might cause subtle symptoms (e.g., fatigue), while severe or prolonged deficiencies can lead to serious conditions (e.g., scurvy from Vitamin C deficiency or beriberi from Vitamin B1 deficiency).

  3. Compounding Effects: Medications depleting multiple nutrients (e.g., corticosteroids affecting calcium, magnesium, and Vitamin D) can lead to compounded symptoms like osteoporosis or muscle dysfunction.


    When things just don't add up, try subtracting...
    When things just don't add up, try subtracting...

 
 
 

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